# Eluxadoline (5-[[[(2S)-2-amino-3-[4-aminocarbonyl)-2,6-dimethylphenyl]-1-oxopropyl][(1S)-1-(4-phenyl-1H-imidazol-2-yl)ethyl]amino]methyl]-2-methoxybenzoic acid) (including its optical isomers) and its salts, isomers, and salts of isomers — Federal controlled substance schedule (I-V) by drug, with DEA code number

For Eluxadoline (5-[[[(2S)-2-amino-3-[4-aminocarbonyl)-2,6-dimethylphenyl]-1-oxopropyl][(1S)-1-(4-phenyl-1H-imidazol-2-yl)ethyl]amino]methyl]-2-methoxybenzoic acid) (including its optical isomers) and its salts, isomers, and salts of isomers, schedule is Schedule IV; listed under is Other substances; dea code number is 9725; cfr citation is 21 CFR 1308.14(g)(3), recorded from its source on 2026-09-01.

- **Substance:** Eluxadoline (5-[[[(2S)-2-amino-3-[4-aminocarbonyl)-2,6-dimethylphenyl]-1-oxopropyl][(1S)-1-(4-phenyl-1H-imidazol-2-yl)ethyl]amino]methyl]-2-methoxybenzoic acid) (including its optical isomers) and its salts, isomers, and salts of isomers _(verified: appears in the quote below)_
- **Schedule:** Schedule IV _(verified: appears in its own passage below)_
- **Listed under:** Other substances _(verified: appears in its own passage below)_
- **DEA code number:** 9725 _(verified: appears in the quote below)_
- **CFR citation:** 21 CFR 1308.14(g)(3) _(our reading, not quoted from the source)_

## What the source says

> (3) Eluxadoline (5-[[[(2S)-2-amino-3-[4-aminocarbonyl)-2,6-dimethylphenyl]-1-oxopropyl][(1S)-1-(4-phenyl-1H-imidazol-2-yl)ethyl]amino]methyl]-2-methoxybenzoic acid) (including its optical isomers) and its salts, isomers, and salts of isomers (9725). |

## Where each value comes from

This source states these in separate places, so each value is shown with the passage that states it.

### Schedule

> § 1308.14 Schedule IV.

### Listed under

> (g) Other substances.

## Source

- https://www.ecfr.gov/current/title-21/chapter-II/part-1308

Last verified: 2026-09-01. Review by: 2026-12-30.
Part of [Federal controlled substance schedule (I-V) by drug, with DEA code number](https://referencesource.org/dea-controlled-substance-schedule-by-drug/).